Discovery of a Highly Selective Sigma-2 Receptor Ligand, 1-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-methyl-1H-b enzo[d]imidazol-2(3H)-one (CM398), with Drug-Like Properties and Antinociceptive Effects In Vivo
Publication Date
7-20-2020
DOI
10.1208/S12248-020-00472-X
ISSN
1550-7416
Recommended Citation
Intagliata, S., Sharma, A., King, T. I., Mesangeau, C., Seminerio, M., Chin, F. T., Wilson, L. L., Matsumoto, R. R., McLaughlin, J. P., Avery, B. A., & McCurdy, C. R. (2020). Discovery of a Highly Selective Sigma-2 Receptor Ligand, 1-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-methyl-1H-b enzo[d]imidazol-2(3H)-one (CM398), with Drug-Like Properties and Antinociceptive Effects In Vivo. AAPS Journal, 22(5), 94. https://doi.org/10.1208/s12248-020-00472-x
PubMed ID
32691179